Discovery of dihydropyridinone derivative as a covalent EZH2 degrader

Bin Zhou(Second Affiliated Hospital of Nanjing Medical University), Aoli Wang(Anhui University), Shuang Qi(People's Liberation Army No. 150 Hospital), Yongfei Chen(Chinese Academy of Sciences), Husheng Mei(University of Science and Technology of China), Wenliang Wang(The University of Texas at Austin), Beilei Wang(Northwestern Polytechnical University), Qingwang Liu(Hefei Institutes of Physical Science), Fengming Zou(Chinese Academy of Sciences), Qingsong Liu(Medical College of Wisconsin), Feiyang Liu(National University of Defense Technology), Rui Jin(Chinese Academy of Sciences), Wenchao Wang(Nanjing Forestry University)
European Journal of Medicinal Chemistry
October 2, 2023
10.1016/j.ejmech.2023.115825
Cited by 11

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