An amide to thioamide substitution improves the permeability and bioavailability of macrocyclic peptides
Pritha Ghosh(Australian National University), Jayanta Chatterjee(Indian Institute of Science Bangalore), Chandrashekar Mataguru Doreswamy(Anthem Biosciences (India)), Nishant Raj(Indian Institute of Science Bangalore), Prem N. Yadav(Punjab Engineering College), Hitesh Verma(Institute of Molecular Biology and Biophysics), Monika Patel(University of Toronto), M. B. Dinesh(Indian Institute of Science Bangalore), Sohini Chakraborti(Institute of Molecular Biology and Biophysics), S. R. Anandakumar(Anthem Biosciences (India)), Srinivas Seekallu(Anthem Biosciences (India)), Gajanan Jadhav(University of Alabama at Birmingham), Bhavesh Khatri(Institute of Molecular Biology and Biophysics)
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