Structure-Based Optimization of Covalent, Small-Molecule Stabilizers of the 14-3-3σ/ERα Protein–Protein Interaction from Nonselective Fragments
Markella Konstantinidou(University of California, San Francisco), Michelle R. Arkin(University of California, San Francisco), Adam R. Renslo(University of California, San Francisco), R. Jeffrey Neitz(University of California, San Francisco), Shubhankar Dutta(University of California, San Francisco), Luc Brunsveld(Eindhoven University of Technology), Edmee Vandenboorn(Eindhoven University of Technology), Maurits Overmans(Eindhoven University of Technology), Sheng Chen(University of California, San Francisco), Christian Ottmann(Max Planck Society), Priyadarshini Jaishankar(University of California, San Francisco), Emira J. Visser(Eindhoven University of Technology)
Cited by 39
Related Papers
Long-Range Photoinduced Electron Transfer Through a DNA Helix
|Science|1993|951
Rates of DNA-Mediated Electron Transfer Between Metallointercalators
|Science|1996|422
First Observation of the Key Intermediate in the “Light-Switch” Mechanism of [Ru(phen)<sub>2</sub>dppz]<sup>2+</sup>
|Journal of the American Chemical Society|1997|375
Covalent inhibitors: a rational approach to drug discovery
|RSC Medicinal Chemistry|2020|375
Fibrin-targeting immunotherapy protects against neuroinflammation and neurodegeneration
|Nature Immunology|2018|210