MCB-613 exploits a collateral sensitivity in drug resistant <i>EGFR</i> -mutant non-small cell lung cancer through covalent inhibition of KEAP1

Christopher F. Bassil(Duke University), Kris C. Wood(Duke University), Kévin Jubien-Girard(Centre National de la Recherche Scientifique), Tierney M. Hall(Duke University), Cécile Favreau(Inserm), Anthony R. Martin(École Nationale Supérieure de Chimie de Montpellier), Haley M. Hutchinson(Duke University), Katherine R. Singleton(Duke University), Shane T. Killarney(Duke University), Christian Cerda-Smith(Duke University), Alexandre Puissant(Délégation Paris 5), Patrick Auberger(Inserm), Guillaume Robert(Centre Méditerranéen de Médecine Moléculaire), Kayleigh N. Askin(Duke University), Rachid Benhida(Centre National de la Recherche Scientifique), Ann Marie Pendergast(Duke University), Peter Winter(Duke University), David M. Lonard(Baylor College of Medicine), Jacob P. Hoj(Duke University), Grace R. Anderson(Duke University), Samuel H. Gruber(Duke University), Li Qin(Baylor College of Medicine), Benjamin Mayro(Duke University)
bioRxiv (Cold Spring Harbor Laboratory)
January 19, 2023
Cited by 0


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