Discovery of (<i>R</i>)-<i>N</i>-Benzyl-2-(2,5-dioxopyrrolidin-1-yl)propanamide [<b>(<i>R</i>)-AS-1</b>], a Novel Orally Bioavailable EAAT2 Modulator with Drug-like Properties and Potent Antiseizure Activity <i>In Vivo</i>

Michał Abram(Jagiellonian University), Krzysztof Kamiński(Jagiellonian University)
Journal of Medicinal Chemistry
August 19, 2022
10.1021/acs.jmedchem.2c00534
Cited by 22

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