Structure-based rational design enables efficient discovery of a new selective and potent AKT PROTAC degrader

Cheng‐Liang Zhu(Zhejiang Lab), Xiaomin Luo(Nanjing University of Chinese Medicine), Tian Tian(Zhejiang University), Zijian Rao(Zhejiang University), Hanlin Wang(Fudan University), Zhesheng Zhou(Zhejiang University), Tian Mi(Shanghai Institute of Materia Medica), Danni Chen(Zhejiang University), Yongjin Xu(Zhejiang Cancer Hospital), Yizhe Wu(Zhejiang University), Jinxin Che(Zhejiang University), Yubo Zhou(Nanjing University of Chinese Medicine), Jia Li(Nanjing University of Chinese Medicine), Xiaowu Dong(Zhejiang Lab)
European Journal of Medicinal Chemistry
May 19, 2022
Cited by 26

Abstract


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