Synthesis of amide and sulfonamide substituted N-aryl 6-aminoquinoxalines as PFKFB3 inhibitors with improved physicochemical properties
Nicolas Boutard, Charles‐Henry Fabritius, Łukasz Włoszczak, Magdalena Sieprawska‐Lupa, Anna Buda, Mirek Jurzak(Merck KGaA, Darmstadt (Germany)), K. Banaszak, Tomasz Rzymski, Sylwia Ziemiańska, Marta Sowińska, Krzysztof Jakubiec, Aleksandra Sabiniarz, Agata Stachowicz, Krzysztof Brzózka, Paulina Niedziejko, Alicja Obara, Marcin Leś, Katarzyna Kwiecińska, Barbara Bugaj, Agata Kitlińska, Ewelina Cieluch, Anna Cierpich, Henryk Pawlik, Marcin Bień, Monika Maciuszek, Artur Biela(Jagiellonian University), Maciej Kujawa, Hans‐Michael Eggenweiler(Merck KGaA, Darmstadt (Germany)), Mateusz M. Tomczyk, Łukasz Dudek, Monika Gaik, Andrzej Gondela, Joanna Fogt, Ralph K. Lindemann(Merck KGaA, Darmstadt (Germany)), Katarzyna Wiklik, Joanna Szeremeta‐Spisak, Piotr Kowalczyk, Mateusz Nowak(The Wojciech Kętrzyński Northern Institute), Paweł Guzik, Adrian Zarębski(Jagiellonian University), Arkadiusz Białas, Maciej Mikulski
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