Identification of Two Non-Peptidergic Small Molecule Inhibitors of CBX2 Binding to K27 Trimethylated Oligonucleosomes

Lukas Lercher(University of Oxford), Michael Finley(Janssen (United States)), Tarig Bashir, Nina Simon(University of Oslo), Torsten Neuefeind, Aaron Patrick(Janssen (United States)), Daniel Riley(Janssen (United States)), Brent Rupnow(Springhouse), Sujata Sharma(Janssen (United States)), David Bochmann, Peter J. Tummino(Intarcia Therapeutics (United States)), Ruth Steele(Janssen (United States)), Vineet Pande(Universidade do Porto), Paul J. Krawczuk(Janssen (United States)), Weixue Wang(Scorpion Therapeutics (United States)), Ben Danna(Janssen (United States)), Andreas Bergmann(MerLion Pharma (Germany)), Marcel J Tauchert
SLAS DISCOVERY
May 2, 2022
Cited by 7


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