Discovery of novel potent covalent inhibitor-based EGFR degrader with excellent in vivo efficacy

Shi Shi(South China Agricultural University), Qihua Zhu(China Pharmaceutical University), Jing Niu(China Pharmaceutical University), Lei Huang(Therapeutics Clinical Research), Yungen Xu(China Pharmaceutical University), Yu Du(China Pharmaceutical University), Jiaqi Cui(China Pharmaceutical University)
Bioorganic Chemistry
January 10, 2022
Cited by 65


Related Papers