Bicyclic Picomolar OGA Inhibitors Enable Chemoproteomic Mapping of Its Endogenous Post-translational Modifications

Manuel González‐Cuesta(Universidad de Sevilla), David J. Vocadlo(Simon Fraser University), Zarina Madden(Simon Fraser University), Alexandra Males(University of York), Roger A. Ashmus(Simon Fraser University), Jason C. Rogalski(University of British Columbia), Cameron Proceviat(Simon Fraser University), Leonard J. Foster(University of British Columbia), Peter Sidhu(University of British Columbia), Carmen Ortiz Mellet(Universidad de Sevilla), José M. Garcı́a Fernández(Centre National de la Recherche Scientifique), Jil A. Busmann(Simon Fraser University), G.J. Davies(New York Structural Biology Center)
Journal of the American Chemical Society
January 5, 2022
Cited by 27


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