Noncovalent CDK12/13 dual inhibitors-based PROTACs degrade CDK12-Cyclin K complex and induce synthetic lethality with PARP inhibitor

Tian Niu(Zhejiang University), Kailin Li(Zhejiang University), Jiang Li(Zhejiang University), Zhesheng Zhou(Zhejiang University), Ju-Eun Hong(Zhejiang University), Xuankun Chen(Zhejiang University), Xiaowu Dong(Zhejiang Lab), Qiaojun He(Zhejiang Lab), Ji Cao(Zhejiang Lab), Bo Yang(Zhejiang University), Cheng‐Liang Zhu(Zhejiang Lab)
European Journal of Medicinal Chemistry
November 25, 2021
Cited by 77Open Access
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