Discovery of <i>N</i>-((3<i>S</i>,4<i>S</i>)-4-(3,4-Difluorophenyl)piperidin-3-yl)-2-fluoro-4-(1-methyl-1<i>H</i>-pyrazol-5-yl)benzamide (Hu7691), a Potent and Selective Akt Inhibitor That Enables Decrease of Cutaneous Toxicity

Jinxin Che(Pharmaceutical Biotechnology (Czechia)), Xiaowu Dong(Second Affiliated Hospital of Zhejiang University), Haichao Sheng(Zhejiang University), Zizheng Gao(Zhejiang University), Bo Yang(Tongde Hospital of Zhejiang Province), Jian Gao(Hebei Medical University), Qinjie Weng(ZheJiang Institute For Food and Drug Control), Peihua Luo(Zhejiang Lab), Zegao Jin(Zhejiang University), Wenhu Zhan(Cornell University), Dan Li(Zhejiang University), Yang Lu(Wuhan University), Qiaojun He(Zhejiang Lab), Yongzhou Hu(Zhejiang University), Xiaoyang Dai(Zhejiang Lab), Binhui Chen(Zhejiang University)
Journal of Medicinal Chemistry
August 10, 2021
Cited by 23


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