Design and Synthesis of EZH2-Based PROTACs to Degrade the PRC2 Complex for Targeting the Noncatalytic Activity of EZH2

Zhihao Liu(Sichuan University), Luoting Yu(State Key Laboratory of Biotherapy), Ningyu Wang(Southwest Jiaotong University), Rong Hu(China Pharmaceutical University), Xingping Su(Sichuan University), Qiangsheng Zhang(Sichuan University), Wei Wei(State Key Laboratory of Biotherapy), Qiwei Wang(Sichuan University), Yongxia Zhu(University of Electronic Science and Technology of China), Hualong He(Sichuan University), Xi Hu(Sichuan University), Tinghong Ye(State Key Laboratory of Biotherapy), Shuyan Zhou(Sichuan University), Xiuli Wu(Sichuan University)
Journal of Medicinal Chemistry
February 19, 2021
Cited by 116


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