Tethered agonist exposure in intact adhesion/class B2 GPCRs through intrinsic structural flexibility of the GAIN domain

Gerti Beliu(University of Würzburg), Steffen Altrichter(Leipzig University), Ramón Guixà-González(Paul Scherrer Institute), Mareike Hemberger(Leipzig University), Ina Brauer(Leipzig University), Anne-Kristin Dahse(Leipzig University), Nicole Scholz(Leipzig University), Robert Wieduwild(Leipzig University), Alexander Kuhlemann(University of Würzburg), Hossein Batebi(Leipzig University), Florian Seufert(Leipzig University), Guillermo Pérez‐Hernández(Charité - Universitätsmedizin Berlin), Peter W. Hildebrand(Berlin Institute of Health at Charité - Universitätsmedizin Berlin), Markus Sauer(University of Würzburg), Tobias Langenhan(Leipzig University)
Molecular Cell
January 25, 2021
Cited by 84

Abstract


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