Discovery of a first-in-class EZH2 selective degrader

Anqi Ma(Icahn School of Medicine at Mount Sinai), Ηλίας Στρατικόπουλος(Icahn School of Medicine at Mount Sinai), Kwang‐Su Park(Icahn School of Medicine at Mount Sinai), Jieli Wei(Icahn School of Medicine at Mount Sinai), Tiphaine Martin(Icahn School of Medicine at Mount Sinai), Xiaobao Yang(Icahn School of Medicine at Mount Sinai), Megan Schwarz(Icahn School of Medicine at Mount Sinai), Violetta V. Leshchenko(Icahn School of Medicine at Mount Sinai), Alexander Rialdi(Icahn School of Medicine at Mount Sinai), Brandon Dale(Icahn School of Medicine at Mount Sinai), Alessandro Laganà(Icahn School of Medicine at Mount Sinai), Ernesto Guccione(Icahn School of Medicine at Mount Sinai), Samir Parekh(Icahn School of Medicine at Mount Sinai), Ramon Parsons(Tisch Hospital), Jian Jin(Icahn School of Medicine at Mount Sinai)
Nature Chemical Biology
December 9, 2019
Cited by 226Open Access
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