Antibody Conjugation of a Chimeric BET Degrader Enables <i>in vivo</i> Activity
Thomas H. Pillow(Genesys (United States)), Peter S. Dragovich(Pfizer (United States)), Shang‐Fan Yu(Genesys (United States)), Tracy Kleinheinz(Genesys (United States)), Brandon Latifi(Genesys (United States)), Isabel Figueroa(Merck & Co., Inc., Rahway, NJ, USA (United States)), Karen E. Gascoigne(University of Manchester), Jack Sadowsky(Genesys (United States)), Cong Wu(Fujian University of Traditional Chinese Medicine), Chun Sing Li(WuXi AppTec (China)), Rebecca K. Rowntree(Genesys (United States)), Donglu Zhang(Acentech (United States)), Pragya Adhikari(Genesys (United States)), Douglas D. Leipold(Genesys (United States)), Katherine R. Kozak(University of California, Los Angeles), Gauri Deshmukh(Yashwantrao Chavan Maharashtra Open University), Zijin Xu(WuXi AppTec (China)), Aimee O’Donohue(Genesys (United States)), Amrita V. Kamath(Bristol-Myers Squibb (United States)), Hongyan Zhang(Tianjin University), Xinxin Wang(Handan College), Jinhua Chen(Hunan University), Hui Yao(Jinan University), Xiaoyu Zhu(WuXi AppTec (China)), Hao Zhou(Institute of Chemical Industry of Forest Products), Ruina Li(Genesys (United States)), Susan Kaufman(Genesys (United States)), Robert A. Blake(Exelixis (United States)), John Wai(WuXi AppTec (China)), Richard Zang(Genesys (United States)), Geoffrey Del Rosario(Genesys (United States)), Melinda M. Mulvihill(Genesys (United States))
Cited by 193
Related Papers
Validation of the ITS2 Region as a Novel DNA Barcode for Identifying Medicinal Plant Species
|PLoS ONE|2010|1.7k
Site-specific conjugation of a cytotoxic drug to an antibody improves the therapeutic index
|Nature Biotechnology|2008|1.4k
Use of ITS2 Region as the Universal DNA Barcode for Plants and Animals
|PLoS ONE|2010|1.2k
Conjugation site modulates the in vivo stability and therapeutic activity of antibody-drug conjugates
|Nature Biotechnology|2012|997