Discovery of piperidine-substituted thiazolo[5,4-d]pyrimidine derivatives as potent and orally bioavailable HIV-1 non-nucleoside reverse transcriptase inhibitors

Dongwei Kang(Shandong University), Xinyong Liu(Shandong University of Traditional Chinese Medicine), Boshi Huang(Virginia Commonwealth University), Christophe Pannecouque(Rega Institute for Medical Research), Erik De Clercq(Rega Institute for Medical Research), Gaochan Wu(Shandong University), Xiaofang Zuo(Shandong University), Fenju Wei(Shandong University), Zhongxia Zhou(Shandong University), Peng Zhan(Shandong University of Traditional Chinese Medicine), Jacob Kongsted(University of Southern Denmark), Heng Zhang(Shandong University), Zhao Wang(Shandong University), Ye Tian(Jilin University), Da Feng(Shandong University), Lanlan Jing(Shandong University), Tong Zhao(China Pharmaceutical University), Vasanthanathan Poongavanam(University of Southern Denmark)
Communications Chemistry
June 28, 2019
Cited by 32


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