Synthesis of (R,S)-isoproterenol, an inhibitor of tau aggregation, as an 11C-labeled PET tracer via reductive alkylation of (R,S)-norepinephrine with [2-11C]acetone

Hiroshi Ikenuma(National Center for Geriatrics and Gerontology), Masaaki Suzuki(Nagoya University), Yasuyuki Kimura(National Center for Geriatrics and Gerontology), Aya Ogata(Gifu University of Medical Science), Kengo Ito(National Center for Geriatrics and Gerontology), Takashi Kato(National Center for Geriatrics and Gerontology), Akihiko Takashima(Gakushuin University), Junichiro Abe(National Center for Geriatrics and Gerontology), Naoya Kajino(Gifu University), Hiroko Koyama(National Center for Geriatrics and Gerontology), Yasuhiro Kawasumi
Bioorganic & Medicinal Chemistry Letters
July 3, 2019
Cited by 5


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