Optimization of the first small-molecule relaxin/insulin-like family peptide receptor (RXFP1) agonists: Activation results in an antifibrotic gene expression profile

Kenneth J. Wilson(National Institutes of Health), Juan Marugán(National Institutes of Health), Emmett R. George(National Institutes of Health), Wei Zheng(Liaoning Cancer Hospital & Institute), Noel Southall(National Institutes of Health), Irina U. Agoulnik(University of South Florida), Alexander I. Agoulnik(Florida International University), Elena Barnaeva(National Center for Advancing Translational Sciences), Xin Hu(Discovery Institute), Amy Wang(National Institutes of Health), Xin Xu(National Institutes of Health), Zaohua Huang(Florida International University), Jingbo Xiao(National Center for Advancing Translational Sciences), Marc Ferrer(National Institute of Biomedical Innovation, Health and Nutrition), Courtney Myhr(Florida International University), Catherine Z. Chen(National Institutes of Health)
European Journal of Medicinal Chemistry
June 7, 2018
Cited by 17


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