Design and synthesis of 4-(2,3-dihydro-1H-benzo[d]pyrrolo[1,2-a]imidazol-7-yl)-N-(5-(piperazin-1-ylmethyl)pyridine-2-yl)pyrimidin-2-amine as a highly potent and selective cyclin-dependent kinases 4 and 6 inhibitors and the discovery of structure-activity relationships

Yan Wang(Capital Medical University), Zhigang Li(Chongqing Medical University), Dianxi Zhu(Jingdong (China)), Heng Li(Central South University), Zhenhua Chen(Jinzhou Medical University), Peng Song(Beijing University of Technology), Lei Yin(Fujian Medical University), Xiu‐Qing Song(Beijing University of Technology), Wenjian Liu(Shandong University), Zhan Wang(Zhejiang Lab), Zhenzhen Cheng(Hunan University)
Bioorganic & Medicinal Chemistry Letters
January 30, 2018
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