Design and synthesis of 4-(2,3-dihydro-1H-benzo[d]pyrrolo[1,2-a]imidazol-7-yl)-N-(5-(piperazin-1-ylmethyl)pyridine-2-yl)pyrimidin-2-amine as a highly potent and selective cyclin-dependent kinases 4 and 6 inhibitors and the discovery of structure-activity relationships

Yan Wang(China Medical University), Zhigang Li(University of Pittsburgh), Dianxi Zhu(Jingdong (China)), Heng Li(Anhui Provincial Hospital), Zhenhua Chen(Jinzhou Medical University), Peng Song(Nanjing Agricultural University), Lei Yin(Jingdong (China)), Xiu‐Qing Song(Beijing University of Technology), Wenjian Liu(Shandong First Medical University), Zhan Wang(Qinghai University), Zhenzhen Cheng(Hunan University)
Bioorganic & Medicinal Chemistry Letters
January 30, 2018
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