Improved Total Synthesis of Tubulysins and Design, Synthesis, and Biological Evaluation of New Tubulysins with Highly Potent Cytotoxicities against Cancer Cells as Potential Payloads for Antibody–Drug Conjugates

K. C. Nicolaou(University of Pennsylvania), Julia Gavrilyuk(Bristol-Myers Squibb (Germany)), Rohan D. Erande(Indian Institute of Technology Jodhpur), Monette Aujay(ChemoCentryx (United States)), Joseph Sandoval(ChemoCentryx (United States)), Stefan Munneke(AbbVie (United States)), Dionisios Vourloumis(Scripps Research Institute), Jun Yin(Central China Normal University)
Journal of the American Chemical Society
January 30, 2018
Cited by 50


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