Allenamide as a bioisostere of acrylamide in the design and synthesis of targeted covalent inhibitorsDeheng Chen(Chinese Academy of Sciences), Yujun Zhao(Chinese Academy of Sciences)MedChemCommDecember 11, 201710.1039/c7md00571gCited by 28SaveCiteExport RISWatch citationsRelated PapersPharmacological blockade of PCAF ameliorates osteoarthritis development via dual inhibition of TNF-α-driven inflammation and ER stress|EBioMedicine|2019|56Structure-Based Discovery of 4-(6-Methoxy-2-methyl-4-(quinolin-4-yl)-9<i>H</i>-pyrimido[4,5-<i>b</i>]indol-7-yl)-3,5-dimethylisoxazole (CD161) as a Potent and Orally Bioavailable BET Bromodomain Inhibitor|Journal of Medicinal Chemistry|2017|42