Lessons in PROTAC Design from Selective Degradation with a Promiscuous Warhead

Daniel P. Bondeson(Yale University), Blake E. Smith(Yale University), George M. Burslem(Yale University), Alexandru D. Buhimschi(Yale University), John Hines(Yale University), Saul Jaime‐Figueroa(Yale University), Jing Wang(Arvinas (United States)), Brian D. Hamman(Arvinas (United States)), Alexey Ishchenko(Arvinas (United States)), Craig M. Crews(Yale University)
Cell chemical biology
November 9, 2017
Cited by 894Open Access
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