Design, synthesis and biological activity of 3-pyrazine-2-yl-oxazolidin-2-ones as novel, potent and selective inhibitors of mutant isocitrate dehydrogenase 1

Tianfang Ma(China Pharmaceutical University), Xiaoming Zha(China Pharmaceutical University), Andreas von Deimling(Heidelberg University), Qihua Zhu(China Pharmaceutical University), Yueqing Gu(China Pharmaceutical University), Stefan Pusch(German Cancer Research Center), Yungen Xu(China Pharmaceutical University), Lijun Yang(Chinese Academy of Medical Sciences & Peking Union Medical College), Fangxia Zou(China Pharmaceutical University)
Bioorganic & Medicinal Chemistry
October 14, 2017
Cited by 14


Related Papers