Identification of a Novel 1,2,3,4-Tetrahydrobenzo[<i>b</i>][1,6]naphthyridine Analogue as a Potent Phosphodiesterase 5 Inhibitor with Improved Aqueous Solubility for the Treatment of Alzheimer’s Disease

Jole Fiorito(Columbia University), Donald W. Landry, Agnieszka Staniszewski(Columbia University), Faisal Saeed(Columbia University), Ottavio Arancio(Columbia University Irving Medical Center), Shijun Yan(University of California, Irvine), Hong Zhang(Columbia University), Shi‐Xian Deng(Columbia University), Jérémie Vendôme(Schrodinger (United States))
Journal of Medicinal Chemistry
October 6, 2017
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