BET protein proteolysis targeting chimera (PROTAC) exerts potent lethal activity against mantle cell lymphoma cells

Baohua Sun; Warren Fiskus; Yimin Qian; Kimal Rajapakshe; Kanak Raina; Kevin Coleman; Andrew P. Crew; Angela Shen; Dyana T. Saenz; Christopher P. Mill; Agnieszka Nowak; Neeraj Jain; L Zhang; M Wang; Joseph D. Khoury; Cristian Coarfa; Craig M. Crews; Kapil N. Bhalla

doi:10.1038/leu.2017.207

BET protein proteolysis targeting chimera (PROTAC) exerts potent lethal activity against mantle cell lymphoma cells

Baohua Sun(The University of Texas MD Anderson Cancer Center), Warren Fiskus(The University of Texas MD Anderson Cancer Center), Yimin Qian(Arvinas (United States)), Kimal Rajapakshe(Baylor College of Medicine), Kanak Raina(Arvinas (United States)), Kevin Coleman(Arvinas (United States)), Andrew P. Crew(Arvinas (United States)), Angela Shen(Arvinas (United States)), Dyana T. Saenz(The University of Texas MD Anderson Cancer Center), Christopher P. Mill(The University of Texas MD Anderson Cancer Center), Agnieszka Nowak(The University of Texas MD Anderson Cancer Center), Neeraj Jain(The University of Texas MD Anderson Cancer Center), L Zhang(The University of Texas MD Anderson Cancer Center), M Wang(The University of Texas MD Anderson Cancer Center), Joseph D. Khoury(The University of Texas MD Anderson Cancer Center), Cristian Coarfa(Baylor College of Medicine), Craig M. Crews(Yale University), Kapil N. Bhalla(The University of Texas MD Anderson Cancer Center)

Leukemia

June 30, 2017

10.1038/leu.2017.207

Cited by 178Open Access

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