Fatty Acid Cysteamine Conjugates as Novel and Potent Autophagy Activators That Enhance the Correction of Misfolded F508del-Cystic Fibrosis Transmembrane Conductance Regulator (CFTR)

Chi B. Vu(Catabasis Pharmaceuticals (United States)), Feng Liu(Fujian Medical University), Antonio E. Lacerda(Charles River Laboratories (United States)), Robert J. Bridges(Rosalind Franklin University of Medicine and Science), Curtis Bordwell(Charles River Laboratories (United States)), Pallavi Lonkar(Wave Life Sciences (United States)), Amal Ting(Catabasis Pharmaceuticals (United States)), Cecilia Peña‐Rasgado(Rosalind Franklin University of Medicine and Science), Dominic Picarella(Millennium Engineering and Integration (United States)), Andrew J. Nichols(New Frontier), Abby L. Sewell(Charles River Laboratories (United States)), Maisy Yeager(Catabasis Pharmaceuticals (United States)), Allison M. Wensley(Catabasis Pharmaceuticals (United States)), Sachin Chandran(Catabasis Pharmaceuticals (United States))
Journal of Medicinal Chemistry
December 15, 2016
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