Covalent targeting of remote cysteine residues to develop CDK12 and CDK13 inhibitors

Tinghu Zhang(Harvard University), Nicholas Kwiatkowski(Harvard University), Calla M Olson(Harvard University), Sarah E. Dixon-Clarke(University of Oxford), Brian J. Abraham(Whitehead Institute for Biomedical Research), Ann Katrin Greifenberg(University of Bonn), Scott B. Ficarro(Boston University), Jonathan M. Elkins(University of Oxford), Yanke Liang(Harvard University), Nancy M. Hannett(Whitehead Institute for Biomedical Research), Theresa Manz(Dana-Farber Cancer Institute), Mingfeng Hao(Harvard University), Bartlomiej Bartkowiak(Duke Medical Center), Arno L. Greenleaf(Duke Medical Center), Jarrod A. Marto(Boston University), Matthias Geyer(University of Bonn), Alex N. Bullock(University of Oxford), Richard A. Young(Whitehead Institute for Biomedical Research), Nathanael S. Gray(Harvard University)
Nature Chemical Biology
August 29, 2016
Cited by 371Open Access
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