Synthesis and Preclinical Evaluation of 2-(2-Furanyl)-7-[2-[4-[4-(2-[<sup>11</sup>C]methoxyethoxy)phenyl]-1-piperazinyl]ethyl]7<i>H</i>-pyrazolo[4,3-<i>e</i>][1,2,4]triazolo[1,5-<i>c</i>]pyrimidine-5-amine ([<sup>11</sup>C]Preladenant) as a PET Tracer for the Imaging of Cerebral Adenosine A<sub>2A</sub> Receptors

Xiaoyun Zhou(University Medical Center Groningen), Philip H. Elsinga(University Medical Center Groningen), Rudi Dierckx(University Medical Center Groningen), Aren van Waarde(University Medical Center Groningen), Shivashankar Khanapur(University Medical Center Groningen), Anja P. Huizing(University Medical Center Groningen), Rolf Zijlma(University Medical Center Groningen), Marianne Schepers(University Medical Center Groningen), Erik F. J. de Vries(University Medical Center Groningen)
Journal of Medicinal Chemistry
October 3, 2014
Cited by 34


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