Discovery and Preclinical Evaluation of BMS-711939, an Oxybenzylglycine Based PPARα Selective Agonist

Yan Shi(Institut des Maladies Métaboliques et Cardiovasculaires), Joseph A. Tino(Institut des Maladies Métaboliques et Cardiovasculaires), Lori Kunselman(Bristol-Myers Squibb (United States)), Henry Ν. C. Wong(Chinese University of Hong Kong), Bang‐Chi Chen(Bristol-Myers Squibb (United States)), Shiwei Tao(Bristol-Myers Squibb (Germany)), Peter T. W. Cheng(Bristol-Myers Squibb (United States)), Michael Cap, Carrie Xu, Michael A. Blanar(Bristol-Myers Squibb (United States)), Rongan Zhang(Bristol-Myers Squibb (United States)), Ngiap‐Kie Lim, Bowman Miao(Louisville Metabolic and Atherosclerosis Research Center), Andrés S. Hernández(Institut des Maladies Métaboliques et Cardiovasculaires), Lawrence J. Kennedy(Bristol-Myers Squibb (United States)), Lisa Zhang(The University of Sydney), Pathanjali Kadiyala(Louisville Metabolic and Atherosclerosis Research Center), Stanley R. Krystek(Collaborative Drug Discovery (United States)), Juliang Zhu(Bristol-Myers Squibb (Germany)), Robert Zahler(Institut des Maladies Métaboliques et Cardiovasculaires), Debra Search(Louisville Metabolic and Atherosclerosis Research Center), J.K. Muckelbauer(Institute of Crystallography), Ranjan Mukherjee(Ligand Pharmaceuticals (United States)), Vinayak Hosagrahara, Hossain Monshizadegan(Louisville Metabolic and Atherosclerosis Research Center), Kenneth T. Locke(Medicines Evaluation Unit), Jun Li(Bristol-Myers Squibb (United States)), Yixin Li(Baylor College of Medicine), Huiping Zhang(Huazhong University of Science and Technology), Litao Zhang(Tianjin University of Traditional Chinese Medicine), Sean Chen(Rutgers, The State University of New Jersey), Rai Ajit K. Srivastava(Drexel University), Ashok K. Trehan(Bristol-Myers Squibb (Germany)), Kevin O’Malley(Medicines Evaluation Unit), ChiehYing Y. Chang(Institute of Crystallography), Zhi Lai(Institut des Maladies Métaboliques et Cardiovasculaires), Thomas Harrity(Bristol-Myers Squibb (United States)), Daniel S. Meyers(Louisville Metabolic and Atherosclerosis Research Center), Denise Grimm(Louisville Metabolic and Atherosclerosis Research Center)
ACS Medicinal Chemistry Letters
April 4, 2016
Cited by 6


Related Papers