8-Substituted Pyrido[3,4-<i>d</i>]pyrimidin-4(3<i>H</i>)-one Derivatives As Potent, Cell Permeable, KDM4 (JMJD2) and KDM5 (JARID1) Histone Lysine Demethylase Inhibitors

Vassilios Bavetsias(Cancer Research UK), Julian Blagg(Altrincham Hospital)
Journal of Medicinal Chemistry
January 7, 2016
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