Kinesin spindle protein (KSP) inhibitors. Part 3: Synthesis and evaluation of phenolic 2,4-diaryl-2,5-dihydropyrroles with reduced hERG binding and employment of a phosphate prodrug strategy for aqueous solubility
R. M. Garbaccio(Merck & Co., Inc., Rahway, NJ, USA (United States)), George D. Hartman(United States Military Academy), Hans E. Huber(United States Military Academy), Edward S. Tasber(United States Military Academy), David Heimbrook(United States Military Academy), Thomayant Prueksaritanont(United States Military Academy), Robert B. Lobell(United States Military Academy), Nancy E. Kohl(United States Military Academy), Kenneth L. Arrington(United States Military Academy), Cathy Shu(United States Military Academy), Kelly Hamilton(United States Military Academy), Eileen S. Walsh(United States Military Academy), Vicki J. South(United States Military Academy), Carolyn A. Buser(United States Military Academy), Maricel Torrent(United States Military Academy), Youwei Yan(United States Military Academy), William F. Hoffman(United States Military Academy), Lawrence C. Kuo(United States Military Academy), Donald E. Slaughter(United States Military Academy), Michael D. Schaber(United States Military Academy), Weikang Tao(Jiangsu Hengrui Medicine (China)), Christy M. Olson(United States Military Academy), Christine Fernandes(United States Military Academy), Mark E. Fraley(United States Military Academy)
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