Kinesin spindle protein (KSP) inhibitors. Part 4: Structure-based design of 5-alkylamino-3,5-diaryl-4,5-dihydropyrazoles as potent, water-soluble inhibitors of the mitotic kinesin KSP
Christopher D. Cox(United States Military Academy), George D. Hartman(Joint BioEnergy Institute), Robert B. Lobell(United States Military Academy), Nancy E. Kohl(United States Military Academy), Kelly Hamilton(United States Military Academy), Eileen S. Walsh(Janssen (Switzerland)), Elizabeth Mahan(United States Military Academy), Vicki J. South(United States Military Academy), Brenda J. Mariano(United States Military Academy), David B. Whitman(United States Military Academy), Carolyn A. Buser(United States Military Academy), Chunze Li(Nanyang Technological University), Bing Lu, Michael J. Breslin(United States Military Academy), Maricel Torrent(United States Military Academy), Youwei Yan(United States Military Academy), Lawrence C. Kuo(United States Military Academy), Donald E. Slaughter(United States Military Academy), Michael D. Schaber(United States Military Academy), Thomayant Prueksaritanont(United States Military Academy), Weikang Tao(Shanghai Medical Information Center), Paul J. Coleman(United States Military Academy)
Cited by 62
Related Papers
Discovery of a selective catalytic p300/CBP inhibitor that targets lineage-specific tumours
|Nature|2017|878
The importance of synthetic chemistry in the pharmaceutical industry
|Science|2019|650
Glioblastoma Eradication Following Immune Checkpoint Blockade in an Orthotopic, Immunocompetent Model
|Cancer Immunology Research|2015|440
Glucuronidation of Statins in Animals and Humans: A Novel Mechanism of Statin Lactonization
|Drug Metabolism and Disposition|2002|346