Discovery of Marinopyrrole A (Maritoclax) as a Selective Mcl-1 Antagonist that Overcomes ABT-737 Resistance by Binding to and Targeting Mcl-1 for Proteasomal Degradation

Kenichiro Doi(Pennsylvania State University), Hong‐Gang Wang(Pennsylvania State University), Wanda Manieri(Moffitt Cancer Center), E. Schönbrunn(Moffitt Cancer Center), Andy Awwad(Penn State Milton S. Hershey Medical Center), Rongshi Li(Moffitt Cancer Center), Shantu Amin(Penn State Milton S. Hershey Medical Center), Thomas P. Loughran(University of Virginia Cancer Center), Gary W. Daughdrill(University of South Florida), Krishne Gowda(Pennsylvania State University), Yan Liu(Carrier (United States)), Xin Liu(Beijing Radiation Center), Hongwei Wu(University of South Florida), Saı̈d M. Sebti(Virginia Commonwealth University), Shen‐Shu Sung(Pennsylvania State University), Alden Dewey(Penn State Milton S. Hershey Medical Center), Chunwei Cheng(Sichuan University), Yong Qin(Sichuan University)
Journal of Biological Chemistry
February 7, 2012
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