Activation of Hsp90 Enzymatic Activity and Conformational Dynamics through Rationally Designed Allosteric Ligands

Sara Sattin(University of Milan), Giorgio Colombo(University of Pavia), Marco Rusnati(Consorzio Interuniversitario per le Biotecnologie), Anna Bernardi(University of Milan), Mike Moses(National Cancer Institute), Marzia Pennati(Fondazione IRCCS Istituto Nazionale dei Tumori), Laura Morelli(University of Milan), Gerolamo Vettoretti(Institute of Chemistry of Molecular Recognition), Alessia Lopergolo(Fondazione IRCCS Istituto Nazionale dei Tumori), Elisabetta Moroni, Thomas L. Prince(National Cancer Institute), Nadia Zaffaroni(Fondazione IRCCS Istituto Nazionale dei Tumori), Abbey D. Zuehlke(National Cancer Institute), Len Neckers(National Institutes of Health), Jiahui Tao(University of California, San Francisco), David A. Agard(University of California, San Francisco), Kristin Beebe(Center for Cancer Research), Toshiki Kijima(Dokkyo Medical University), Antonella Bugatti(University of Brescia)
Chemistry - A European Journal
August 18, 2015
Cited by 70


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