Regio‐ and Enantioselective Aza‐Diels–Alder Reactions of 3‐Vinylindoles: A Concise Synthesis of the Antimalarial Spiroindolone NITD609

Haifeng Zheng(Luliang University), Xiaoming Feng(Chengdu University), Chaoran Xu(Sichuan University), Yong Xia(Chongqing University), Lili Lin(Colorado Department of Public Health and Environment), Xiaohua Liu(Jiangxi Academy of Forestry)
Angewandte Chemie International Edition
July 23, 2015
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