In Vivo Quantification of Calcitonin Gene-Related Peptide Receptor Occupancy by Telcagepant in Rhesus Monkey and Human Brain Using the Positron Emission Tomography Tracer [11C]MK-4232

Eric D. Hostetler(United States Military Academy), Aniket Joshi(Merck & Co., Inc., Rahway, NJ, USA (United States)), Sandra Sanabria Bohórquez(United States Nuclear Regulatory Commission), Hong Fan(Gwynedd Mercy University), Zhizhen Zeng(United States Military Academy), Mona Purcell(United States Military Academy), Liza Gantert(Merck & Co., Inc., Rahway, NJ, USA (United States)), Kerry Riffel(MSD (Belgium)), Mangay Williams(MSD (Belgium)), Stacey O’Malley(United States Military Academy), Patricia Miller(Merck & Co., Inc., Rahway, NJ, USA (United States)), Harold G. Selnick(United States Nuclear Regulatory Commission), Steven N. Gallicchio(United States Nuclear Regulatory Commission), Ian M. Bell(Gwynedd Mercy University), Christopher Salvatore(MSD (Belgium)), Stefanie A. Kane(United States Military Academy), Chi‐Chung Li(KU Leuven), Richard Hargreaves(Merck & Co., Inc., Rahway, NJ, USA (United States)), Tjibbe de Groot(United States Military Academy), Guy Bormans(MSD (Belgium)), Anne Van Hecken(United States Nuclear Regulatory Commission), Inge Derdelinckx(MSD (Belgium)), Jan de Hoon(Merck & Co., Inc., Rahway, NJ, USA (United States)), Tom Reynders(MSD (Belgium)), Ruben Declercq(United States Nuclear Regulatory Commission), Inge De Lepeleire(United States Military Academy), William P. Kennedy(United States Nuclear Regulatory Commission), Rebecca Blanchard(United States Military Academy), Eugene E. Marcantonio(Merck & Co., Inc., Rahway, NJ, USA (United States)), Cyrille Sur(United States Military Academy), Jacquelynn J. Cook(Gwynedd Mercy University), Koen Van Laere(Gwynedd Mercy University), Jeffrey L. Evelhoch(United States Military Academy)
Journal of Pharmacology and Experimental Therapeutics
August 24, 2013
Cited by 129

Abstract


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