A common pharmacophore for epothilone and taxanes: Molecular basis for drug resistance conferred by tubulin mutations in human cancer cells
Paraskevi Giannakakou(Cornell University), Tito Fojo(James J. Peters VA Medical Center), K. C. Nicolaou(Scripps Research Institute), Kenneth H. Downing(University of Louisiana at Lafayette), Dan L. Sackett, Birgit Bollbuck(National Institute of Diabetes and Digestive and Kidney Diseases), Eva Nogales(Howard Hughes Medical Institute), Rick Gussio(National Institute of Diabetes and Digestive and Kidney Diseases), Daniel Zaharevitz(National Institute of Diabetes and Digestive and Kidney Diseases), George Poy(National Institutes of Health)
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