Distinct pharmacology of rat and human histamine H<sub>3</sub> receptors: role of two amino acids in the third transmembrane domain
Xavier Ligneau(Inserm), J Tardivel‐Lacombe(Inserm), Walter Schunack, C. Robin Ganellin(University College London), Florence Gbahou, Séverine Morisset‐Lopez(Centre National de la Recherche Scientifique), Holger Stark(Heinrich Heine University Düsseldorf)
Cited by 149
Related Papers
International Union of Basic and Clinical Pharmacology. XCVIII. Histamine Receptors
|Pharmacological Reviews|2015|558
Polypharmacology by Design: A Medicinal Chemist’s Perspective on Multitargeting Compounds
|Journal of Medicinal Chemistry|2018|476
Attenuation of levodopa-induced dyskinesia by normalizing dopamine D3 receptor function
|Nature Medicine|2003|381
DOGS: Reaction-Driven de novo Design of Bioactive Compounds
|PLoS Computational Biology|2012|264
Neurochemical and Behavioral Effects of Ciproxifan, A Potent Histamine H3-Receptor Antagonist
|Journal of Pharmacology and Experimental Therapeutics|1998|240