Design and chemoproteomic functional characterization of a chemical probe targeted to bromodomains of BET family proteins

Jiang Wu(Pfizer (United States)), Julia Shin(Pfizer (United States)), Cara Williams(Pfizer (United States)), Kieran F. Geoghegan(Pfizer (United States)), Stephen W. Wright(Pfizer (United States)), David C. Limburg(Pfizer (United States)), Parag V. Sahasrabudhe(Pfizer (United States)), Paul D. Bonin(Pfizer (United States)), Bruce A. Lefker(Pfizer (United States)), Simeon Ramsey(Pfizer (United States))
MedChemComm
January 1, 2014
Cited by 11

Abstract

Selectivity of a <bold>PFI-1</bold> based BET bromodomain probe was demonstrated using affinity capture in nuclear extracts from human cells.


Related Papers

No related papers found

Powered by citation graph analysis