Discovery of XL888: A novel tropane-derived small molecule inhibitor of HSP90
Joerg Bussenius(Exelixis (United States)), Charles M. Blazey(Exelixis (United States)), Naing Aay(Exelixis (United States)), Neel K. Anand(Exelixis (United States)), Arlyn Arcalas(Exelixis (United States)), TaeGon Baik(Exelixis (United States)), O.J. Bowles(Exelixis (United States)), Chris A. Buhr(Exelixis (United States)), Simona Costanzo(Exelixis (United States)), Jeffrey K. Curtis(Exelixis (United States)), Steven C. DeFina(Exelixis (United States)), L. G. DUBENKO(Exelixis (United States)), Timothy S. Heuer(Exelixis (United States)), Ping Huang(Exelixis (United States)), Christopher T. Jaeger(Exelixis (United States)), Anagha A. Joshi(Exelixis (United States)), A.R. Kennedy(Exelixis (United States)), Angie I. Kim(Exelixis (United States)), Katherine Lara(Exelixis (United States)), Jae Lee(Exelixis (United States)), Jonathan Li(Exelixis (United States)), Julie C. Lougheed(Exelixis (United States)), Sunghoon Ma(Exelixis (United States)), Shiva Malek(Exelixis (United States)), Jean-Claire L. Manalo(Exelixis (United States)), Jean‐François Martini(Exelixis (United States)), Garth McGrath(Exelixis (United States)), Monique Nicoll(Exelixis (United States)), John M. Nuss(Exelixis (United States)), Michael Pack(Exelixis (United States)), Csaba J. Peto(Exelixis (United States)), Tsze H. Tsang(Exelixis (United States)), Longcheng Wang(Exelixis (United States)), Scott W. Womble(Exelixis (United States)), Michael Yakes(Exelixis (United States)), Wentao Zhang(Exelixis (United States)), Kenneth D. Rice(Exelixis (United States))
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