Spirocyclic ureas: Orally bioavailable 11β-HSD1 inhibitors identified by computer-aided drug design

Colin M. Tice, David A. Claremon, Gerard M. McGeehan, R. David Simpson(Institute of Forest Science), Barbara A. Kruk, Joan Guo, Richard K. Harrison(Tel Aviv University), Jennifer Berbaum, Reshma Panemangalore, Paula M. Krosky, Yuri Bukhtiyarov, Wei Zhao, Suresh B. Singh(Unknown), Brian M. McKeever(Merck & Co., Inc., Rahway, NJ, USA (United States)), Yuan-Jie Ye, Salvacion Cacatian, Wei He(Northeast Agricultural University), Zhenrong Xu(Minzu University of China), Boyd B. Scott, Linghang Zhuang, Judith Johnson, Joseph G. Bruno, Peter Lindblom, Yi Zhao(National University of Singapore)
Bioorganic & Medicinal Chemistry Letters
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