Synthesis and structure–activity relationship of 2-adamantylmethyl tetrazoles as potent and selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1)

Xiang‐Yang Ye(Hangzhou Normal University), Jeffrey A. Robl(Bristol-Myers Squibb (Germany)), Ramakrishna Seethala(Bristol-Myers Squibb (United States)), Rajasree Golla(Bristol-Myers Squibb (United States)), Akbar Nayeem(Bristol-Myers Squibb (United States)), Bogdan Sleczka(Bristol-Myers Squibb (United States)), Bin He(Guiyang Medical University), David Yoon(Bristol-Myers Squibb (United States)), Mengmeng Wang(Bristol-Myers Squibb (United States)), Yixin Li(Qinghai University), Stephanie Chen(Bristol-Myers Squibb (United States)), David A. Gordon(Bristol-Myers Squibb (United States)), Timothy W. Harper(Bristol-Myers Squibb (United States)), Mark Kirby(Bristol-Myers Squibb (United States)), Atsu Apedo(Bristol-Myers Squibb (United States))
Bioorganic & Medicinal Chemistry Letters
December 5, 2013
Cited by 17


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