A potentiator of orthosteric ligand activity at GLP-1R acts via covalent modification

Whitney M. Nolte(Pfizer (United States)), Jean‐Philippe Fortin(Pfizer (United States)), Benjamin D. Stevens(Pfizer (United States)), Gary E. Aspnes(Pfizer (United States)), David A. Griffith(Pfizer (United States)), Lise R. Hoth(Pfizer (United States)), Roger B. Ruggeri(Pfizer (United States)), Alan M. Mathiowetz(Pfizer (United States)), Chris Limberakis(Pfizer (United States)), David Hepworth(Pfizer (United States)), Philip A. Carpino(Pfizer (United States))
Nature Chemical Biology
July 6, 2014
Cited by 87

Abstract


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