Synthesis and structure–activity relationships of dual PI3K/mTOR inhibitors based on a 4-amino-6-methyl-1,3,5-triazine sulfonamide scaffold

Ryan P. Wurz(Amgen (United States)), Mark H. Norman(Amgen (United States)), Nancy R. Zhang(University of the Arts), Nobuko Nishimura(Amgen (United States)), Kevin Yang(Revolution Medicines (United States)), Tisha San Miguel(Amgen (United States)), Douglas A. Whittington(Amgen (United States)), Erin L. Mullady(Amgen (United States)), Liping H. Pettus(Amgen (United States)), Jian Jiang(Xuzhou Medical College), Longbin Liu(National University of Defense Technology), Ling Wang(Guizhou University), Paul E. Hughes(Amgen (United States)), Sean Caenepeel(Amgen (United States)), Kristin L. Andrews(Amgen (United States)), Yunxin Bo(Amgen (United States)), John D. McCarter(Amgen (United States)), Daniel J. Freeman(Amgen (United States)), Raju Subramanian(Gilead Sciences (United States))
Bioorganic & Medicinal Chemistry Letters
July 4, 2012
Cited by 30


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