Design and synthesis of 6-fluoro-2-naphthyl derivatives as novel CCR3 antagonists with reduced CYP2D6 inhibition

Ippei Sato(Astellas Pharma (Japan)), Shin‐ichi Tsukamoto(Astellas Pharma (Japan)), Yosuke Iura(Toray (United States)), Hirokazu Kubota(Astellas Pharma (Japan)), Koichiro Morihira(Astellas Pharma (Japan)), Toshiya Takahashi(Tohoku University), Takayuki Imaoka(Toray Industries, Inc. (Japan)), Tatsuaki Morokata(Astellas Pharma (Japan)), Makoto Takeuchi(Astellas Pharma (Japan)), Hiroshi Inami(Astellas Pharma (Japan)), A. Nitta(Toray (United States)), Mitsuaki Ohta(Tokyo University of Agriculture)
Bioorganic & Medicinal Chemistry
August 8, 2008
Cited by 14


Related Papers