Discovery of the First Potent and Orally Efficacious Agonist of the Orphan G-Protein Coupled Receptor 119

Graeme Semple(Eurofins (United States)), Robert M. Jones(Arena Pharmaceuticals (United States)), Christopher J. Carroll(St George's, University of London), Karoline Choi(Arena Pharmaceuticals (United States)), Charles Xing(Arena Pharmaceuticals (United States)), Michael Morgan(Arena Pharmaceuticals (United States)), Stuart Bossie(Arena Pharmaceuticals (United States)), David J. Unett(Arena Pharmaceuticals (United States)), William Thomsen, Beatriz Fioravanti(Arena Pharmaceuticals (United States)), Imelda Calderon(Arena Pharmaceuticals (United States)), Yifeng Xiong(Collaborative Innovation Center of Advanced Microstructures), Erin K. Hauser(Arena Pharmaceuticals (United States)), Jane Uy(Arena Pharmaceuticals (United States)), Andrew J. Grottick, James Leonard(Arena Pharmaceuticals (United States)), Albert Ren, Guilherme Rocha Pereira(Pontifícia Universidade Católica de Minas Gerais), Vibha Davé(Arena Pharmaceuticals (United States)), Zhi‐Liang Chu(Arena Pharmaceuticals (United States))
Journal of Medicinal Chemistry
August 13, 2008
Cited by 142


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