The 2.5 Å Crystal Structure of the SIRT1 Catalytic Domain Bound to Nicotinamide Adenine Dinucleotide (NAD<sup>+</sup>) and an Indole (EX527 Analogue) Reveals a Novel Mechanism of Histone Deacetylase Inhibition

Xun Zhao(Center Point), J.G. Luz(Center Point), James A. Jamison(Eli Lilly (United States)), Bradley Condon(Center Point), T. Gheyi(Center Point), Marijane Russell(Center Point), Aiping Zhang(Yangzhou University), Dagart Allison(Center Point), S. Ashok(Center Point), Iain MacEwan(University of California San Diego), Feiyu Zhang(Hubei University of Science and Technology), Yuewei Qian(Eli Lilly (United States))
Journal of Medicinal Chemistry
January 11, 2013
Cited by 218


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