Selective inhibition of BET bromodomains

P. Filippakopoulos(University of Oxford), Jun Qi(Dana-Farber Cancer Institute), S. Picaud(University of Oxford), Y. Shen(University of Notre Dame), William Smith(Harvard University), O. Fedorov(University of Oxford), Elizabeth M. Morse(Harvard University), T. Keates(Genomics (United Kingdom)), Tyler Hickman(Harvard University), I. Felletar(University of Oxford), Martin Philpott(University of Oxford), Shonagh Munro(University of Oxford), Michael R. McKeown(Dana-Farber Cancer Institute), Yuchuan Wang(Harvard University), Amanda L. Christie(Harvard University), Nathan West(Harvard University), Michael J. Cameron(Brigham and Women's Hospital), Brian E. Schwartz(Harvard University), Tom D. Heightman(Genomics (United Kingdom)), Nicholas La Thangue(University of Oxford), Christopher A. French(Brigham and Women's Hospital), Olaf Wiest(University of Notre Dame), Andrew L. Kung(Imaging Center), Stefan Knapp(University of Oxford), James E. Bradner(Dana-Farber Cancer Institute)
Nature
September 24, 2010
Cited by 4,280Open Access
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