Conformation-Dependent Ligand Regulation of ATP Hydrolysis by Human KSP: Activation of Basal Hydrolysis and Inhibition of Microtubule-Stimulated Hydrolysis by a Single, Small Molecule Modulator
Lusong Luo(Beijing Biocytogen (China)), Robert A. Copeland(Unknown), Stephen J. Coales(GlaxoSmithKline (United States)), Dashyant Dhanak(Wilmington University), Kathleen S. Molnar(University of California, San Francisco), Peter J. Tummino(Intarcia Therapeutics (United States)), Pearl S. Huang(Merck & Co., Inc., Rahway, NJ, USA (United States)), Yoshitomo Hamuro(GlaxoSmithKline (United States)), Steven Tuske(GlaxoSmithKline (United States)), Jeffrey R. Jackson(New Frontier), Chiu-Mei Sung(South College), Jeffrey D. Carson(GlaxoSmithKline (United States)), Kurt R. Auger(Research Triangle Park Foundation), Valery Sudakin(Technion – Israel Institute of Technology)
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